Tadalafil
FDA-Approved moleculeCompounded form not FDA-approvedAlso known as: Cialis, PDE5 inhibitor
Phosphodiesterase type 5 (PDE5) inhibitor
- How it works
- Blocks the PDE5 enzyme to improve blood flow in erectile tissue; noted for a longer duration of action than sildenafil.
- Known risks
- Headache, back/muscle aches, flushing, indigestion; rare priapism and sudden sensory changes.
- Contraindications
- Concurrent nitrate therapy; certain cardiovascular conditions.
- Drug interactions
- Hypotension with nitrates and alpha-blockers; levels affected by CYP3A4 inhibitors.
Citations
- Efficacy and safety of tadalafil for the treatment of erectile dysfunction (2002) · PMID 12352383
This information is educational only and is not medical advice. A licensed provider makes all clinical decisions. Diadara provides no dosing, reconstitution, or administration guidance.
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